![Utilizing comprehensive and mini-kinome panels to optimize the selectivity of quinoline inhibitors for cyclin G associated kinase (GAK) - ScienceDirect Utilizing comprehensive and mini-kinome panels to optimize the selectivity of quinoline inhibitors for cyclin G associated kinase (GAK) - ScienceDirect](https://ars.els-cdn.com/content/image/1-s2.0-S0960894X19303221-ga1.jpg)
Utilizing comprehensive and mini-kinome panels to optimize the selectivity of quinoline inhibitors for cyclin G associated kinase (GAK) - ScienceDirect
![Clustering analysis of recently approved kinase inhibitors presented at Discovery on Target 2020 - Virtual - Oncolines B.V. Clustering analysis of recently approved kinase inhibitors presented at Discovery on Target 2020 - Virtual - Oncolines B.V.](https://www.oncolines.com/wp-content/uploads/2020/09/NTRC_DoT20_clustering-of-kinase-inhibitors_web.png)
Clustering analysis of recently approved kinase inhibitors presented at Discovery on Target 2020 - Virtual - Oncolines B.V.
![Kinase Selectivity. A: Each compound was profiled against a panel of... | Download Scientific Diagram Kinase Selectivity. A: Each compound was profiled against a panel of... | Download Scientific Diagram](https://www.researchgate.net/profile/Roland-Kontermann/publication/49694914/figure/fig3/AS:305886879862786@1449940523105/Kinase-Selectivity-A-Each-compound-was-profiled-against-a-panel-of-239-protein-kinases_Q640.jpg)
Kinase Selectivity. A: Each compound was profiled against a panel of... | Download Scientific Diagram
![A) KinomeScanTreeSpot description of the 6i selectivity profile. 6i... | Download Scientific Diagram A) KinomeScanTreeSpot description of the 6i selectivity profile. 6i... | Download Scientific Diagram](https://www.researchgate.net/publication/286486943/figure/fig4/AS:639765745520640@1529543448518/A-KinomeScanTreeSpot-description-of-the-6i-selectivity-profile-6i-was-screened-against.png)
A) KinomeScanTreeSpot description of the 6i selectivity profile. 6i... | Download Scientific Diagram
![Comprehensive assay of kinase catalytic activity reveals features of kinase inhibitor selectivity | Nature Biotechnology Comprehensive assay of kinase catalytic activity reveals features of kinase inhibitor selectivity | Nature Biotechnology](https://media.springernature.com/lw685/springer-static/image/art%3A10.1038%2Fnbt.2017/MediaObjects/41587_2011_Article_BFnbt2017_Fig1_HTML.jpg)
Comprehensive assay of kinase catalytic activity reveals features of kinase inhibitor selectivity | Nature Biotechnology
![PKIS deep dive yields a chemical starting point for dark kinases and a cell active BRSK2 inhibitor | Scientific Reports PKIS deep dive yields a chemical starting point for dark kinases and a cell active BRSK2 inhibitor | Scientific Reports](https://media.springernature.com/m685/springer-static/image/art%3A10.1038%2Fs41598-020-72869-9/MediaObjects/41598_2020_72869_Fig1_HTML.png)
PKIS deep dive yields a chemical starting point for dark kinases and a cell active BRSK2 inhibitor | Scientific Reports
![Figure 10, Kinase Panel Screen for ML264 (no significant kinase activity was seen) - Probe Reports from the NIH Molecular Libraries Program - NCBI Bookshelf Figure 10, Kinase Panel Screen for ML264 (no significant kinase activity was seen) - Probe Reports from the NIH Molecular Libraries Program - NCBI Bookshelf](https://www.ncbi.nlm.nih.gov/books/NBK143546/bin/ml264f10.jpg)
Figure 10, Kinase Panel Screen for ML264 (no significant kinase activity was seen) - Probe Reports from the NIH Molecular Libraries Program - NCBI Bookshelf
![ePosters - Bioluminescent Kinase Profiling Systems For Characterizing Small Molecule Kinase Inhibitors ePosters - Bioluminescent Kinase Profiling Systems For Characterizing Small Molecule Kinase Inhibitors](https://www.eposters.net/thumbnails/bioluminescent-kinase-profiling-systems-for-characterizing-small-molecule-kinase-inhibitors.png)
ePosters - Bioluminescent Kinase Profiling Systems For Characterizing Small Molecule Kinase Inhibitors
Receptor Tyrosine Kinases Activate Canonical WNT/β-Catenin Signaling via MAP Kinase/LRP6 Pathway and Direct β-Catenin Phosphorylation | PLOS ONE
![Kinase inhibition profiles as a tool to identify kinases for specific phosphorylation sites | Nature Communications Kinase inhibition profiles as a tool to identify kinases for specific phosphorylation sites | Nature Communications](https://media.springernature.com/full/springer-static/image/art%3A10.1038%2Fs41467-020-15428-0/MediaObjects/41467_2020_15428_Fig1_HTML.png)
Kinase inhibition profiles as a tool to identify kinases for specific phosphorylation sites | Nature Communications
![Bioluminescent kinase strips: A novel approach to targeted and flexible kinase inhibitor profiling - ScienceDirect Bioluminescent kinase strips: A novel approach to targeted and flexible kinase inhibitor profiling - ScienceDirect](https://ars.els-cdn.com/content/image/1-s2.0-S0003269715005333-gr1.jpg)
Bioluminescent kinase strips: A novel approach to targeted and flexible kinase inhibitor profiling - ScienceDirect
![Panel of binding assays for 113 different protein kinases.Each kinase... | Download Scientific Diagram Panel of binding assays for 113 different protein kinases.Each kinase... | Download Scientific Diagram](https://www.researchgate.net/publication/8020753/figure/fig2/AS:317000015466512@1452590101861/Panel-of-binding-assays-for-113-different-protein-kinasesEach-kinase-represented-in-the.png)
Panel of binding assays for 113 different protein kinases.Each kinase... | Download Scientific Diagram
![Kinase Selectivity Profiling Systems (KSPS) assay principle. (A) Kinase... | Download Scientific Diagram Kinase Selectivity Profiling Systems (KSPS) assay principle. (A) Kinase... | Download Scientific Diagram](https://www.researchgate.net/publication/310390993/figure/fig1/AS:429434680418304@1479396614293/Kinase-Selectivity-Profiling-Systems-KSPS-assay-principle-A-Kinase-targets-selected.png)